An efficient method for the preparation of peptide alcohols.
نویسندگان
چکیده
N-protected LL-dipeptide alcohols 3a-p, diastereomeric mixture (3d + 3d') and tripeptide alcohols 6a-c were synthesized by treatment of various amino alcohols with N-protected(alpha-aminoacyl)benzotriazoles 1a-c, 1f-m, (1a + 1a') and N-protected(alpha-dipeptidoyl)benzotriazoles 5a, 5b respectively in good yields with complete retention of chirality.
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ورودعنوان ژورنال:
- Organic & biomolecular chemistry
دوره 7 21 شماره
صفحات -
تاریخ انتشار 2009